Cyclomethycaine

Cyclomethycaine is an ester-type local anesthetic used for surface anesthesia by inhibiting nerve impulse transmission.

Structure of Cyclomethycaine

• It is a synthetic local anesthetic with a cyclohexylmethyl substituent attached to a benzamide core.
• Chemical Formula: C₁₀H₁₈N₂O

Mode of Action

• Voltage-Gated Sodium Channel Blockade: Prevents nerve impulse conduction by inhibiting sodium channels.
• Localized Action: Provides effective local anesthesia with minimal systemic absorption.

Uses

• Ophthalmic Procedures: Used in eye surgeries for corneal anesthesia.
• Dental Anesthesia: Applied in dental procedures for numbing soft tissues.
• Minor Skin Procedures: Used for minor dermatological procedures requiring local numbing.

Side Effects of Cyclomethycaine

• Local Irritation: Redness and mild irritation at the application site.
• Allergic Reactions: Rare but possible in sensitive individuals.

Thank you for reading from Firsthope's notes, don't forget to check YouTube videos!