Diperodon

Diperodon is a local anesthetic applied topically in ophthalmology and dentistry to numb mucous membranes.

Structure of Diperodon

• It is a synthetic amino benzoic acid derivative with a cyclohexylmethyl substituent, enhancing its local anesthetic potency.
• Chemical Formula: C₁₀H₂₀N₂O₂

Mode of Action

• Voltage-Gated Sodium Channel Inhibition: Blocks sodium influx, preventing nerve impulse transmission.
• Membrane Stabilization: Reduces nerve excitability by stabilizing neuronal membranes.

Uses

• Local Anesthesia: Used in dental procedures, minor surgical interventions, and dermatological applications.
• Topical Preparations: Applied to skin and mucous membranes for temporary numbing.
• Ophthalmic Anesthesia: Employed in eye surgeries for effective corneal numbing.

Side Effects of Diperodon

• Local Reactions: Redness, swelling, or irritation at the application site.
• Systemic Toxicity: Potential CNS and cardiovascular effects with excessive use.

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