Diperodon

Diperodon

Diperodon is a local anesthetic applied topically in ophthalmology and dentistry to numb mucous membranes. Structure of Diperodon It is a synthetic amino benzoic acid derivative with a cyclohexylmethyl substituent, enhancing its local anesthetic potency. Chemical Formula: C₁₀H₂₀N₂O₂ Mode of Action Voltage-Gated Sodium Channel Inhibition: Blocks sodium influx, preventing nerve impulse transmission. Membrane Stabilization: Reduces … Read more

Phenacaine

Phenacaine

Phenacaine is an ester-type local anesthetic used mainly in ophthalmology for surface eye anesthesia. Structure of Phenacaine It is an amino benzoic acid derivative with a propyl ester group, providing effective local anesthetic properties. Chemical Formula: C₁₀H₂₀N₂O₂ Mode of Action Sodium Channel Blockade: Inhibits voltage-gated sodium channels, preventing nerve impulse conduction. Membrane Stabilization: Enhances nerve … Read more

Etidocaine

Etidocaine

Etidocaine is a long-acting amide local anesthetic used for surgical anesthesia and nerve blocks. Structure of Etidocaine It is an amide-type local anesthetic with an extended diethylaminoethyl side chain, providing prolonged anesthetic effects. Chemical Formula: C₁₅H₂₈N₂O Mode of Action Sodium Channel Inhibition: Blocks voltage-gated sodium channels, preventing nerve impulse propagation. Membrane Stabilization: Reduces nerve excitability … Read more

Mepivacaine

Mepivacaine

Mepivacaine is an amide local anesthetic used for infiltration and regional anesthesia with rapid onset and moderate duration. Structure of Mepivacaine It is an amide-type local anesthetic similar to lidocaine but with a methyl group attached to the diethylaminoethyl side chain, enhancing its potency. Chemical Formula: C₁₄H₂₈N₂O Mode of Action Sodium Channel Blockade: Blocks voltage-gated … Read more

Piperocaine

Piperocaine

Piperocaine is an ester-type local anesthetic used for infiltration and surface anesthesia by blocking nerve conduction. Structure of Piperocaine It is a synthetic local anesthetic with a piperidine ring attached to a benzamide core, enhancing its anesthetic potency and duration. Chemical Formula: C₁₀H₂₁N₃O Mode of Action Sodium Channel Inhibition: Blocks voltage-gated sodium channels, preventing nerve … Read more

Cyclomethycaine

Cyclomethycaine

Cyclomethycaine is an ester-type local anesthetic used for surface anesthesia by inhibiting nerve impulse transmission. Structure of Cyclomethycaine It is a synthetic local anesthetic with a cyclohexylmethyl substituent attached to a benzamide core. Chemical Formula: C₁₀H₁₈N₂O Mode of Action Voltage-Gated Sodium Channel Blockade: Prevents nerve impulse conduction by inhibiting sodium channels. Localized Action: Provides effective … Read more

Lignocaine

Lignocaine

Lignocaine (Lidocaine) is a widely used amide local anesthetic for infiltration, nerve blocks, and surface anesthesia. Structure of Lignocaine Lignocaine, commonly known as Lidocaine, is an amide-type local anesthetic with a diethylaminoethyl side chain attached to a 1,5-dimethyl-2-phenyl-4-imidazolidinone core. Chemical Formula: C₁₂H₂₁N₃O Mode of Action Voltage-Gated Sodium Channel Blockade: Inhibits sodium influx, preventing nerve impulse … Read more

Benoxinate

Benoxinate

Benoxinate is an ester local anesthetic mainly used in ophthalmology to numb the eye surface for diagnostic procedures. Structure of Benoxinate It is an amino benzoic acid derivative with a butyl ester group, primarily used in ophthalmic preparations for its local anesthetic properties. Chemical Formula: C₁₂H₂₀N₂O₂ Mode of Action Sodium Channel Inhibition: Blocks voltage-gated sodium … Read more

Tetracaine

Tetracaine

Tetracaine is a potent ester local anesthetic used for spinal and ophthalmic anesthesia by blocking nerve signals. Structure of Tetracaine It is a potent amino benzoic acid derivative with a butyl ester group, providing long-lasting local anesthetic effects. Chemical Formula: C₁₂H₂₉N₃O₂ Mode of Action Sodium Channel Blockade: Inhibits voltage-gated sodium channels, preventing nerve impulse conduction. … Read more

Propoxycaine

Propoxycaine

Propoxycaine is an ester-type local anesthetic used with procaine for dental procedures by blocking nerve conduction. Structure of Propoxycaine It is an amino benzoic acid derivative with a propoxyethyl ester group, enhancing its solubility and anesthetic efficacy. Chemical Formula: C₁₂H₂₉N₃O₂ Mode of Action Sodium Channel Inhibition: Blocks voltage-gated sodium channels, preventing nerve impulse transmission. Membrane … Read more