- Ethchlorvynol acts on the CNS, enhancing inhibitory pathways to induce sleep and relaxation.
- It is used as a sedative-hypnotic for short-term relief of insomnia.
Chemical Formula:
- C₇H₁₁ClO
Mechanism of Action:
- CNS depressant with barbiturate-like action
- Potentiates GABA-mediated chloride currents
Therapeutic Uses of Ethchlorvynol:
- Insomnia (short-term)
Side Effects of Ethchlorvynol:
- Dizziness
- Euphoria
- Nausea
- Risk of dependence, delirium, or psychosis (at high doses)
SAR Notes:
- Lipophilic alcohol core enhances CNS penetration.
- Chlorine and vinyl substitutions increase potency.
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